SCHEMBL485998

SCHEMBL485998

CC(O)c1nc2ccccc2s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.64
LOXL2 Q9Y4K0 1/20 0.62
TSHR P16473 2/20 0.56
GAA P10253 2/20 0.56
ALOX5 P09917 1/20 0.56
MAPK1 P28482 1/20 0.56
HSD17B10 Q99714 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
HIF1A Q16665 1/20 0.54
CASR P41180 1/20 0.53
RAB9A P51151 3/20 0.51
ALOX15 P16050 2/20 0.49
CASP1 P29466 1/20 0.49
MAPT P10636 2/20 0.47
PAX8 Q06710 1/20 0.47
NOD2 Q9HC29 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
APEX1 P27695 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17947424 1.00 HPGD (0.64) HPGDLOXL2TSHRGAAALOX5
SCHEMBL12085830 1.00 HPGD (0.64) HPGDLOXL2TSHRGAAALOX5
SCHEMBL2146969 0.84 LOXL2 (0.66) HPGDLOXL2TSHRGAAALOX5
SCHEMBL62420 0.84 LOXL2 (0.66) HPGDLOXL2TSHRGAAALOX5
SCHEMBL9675088 0.82 LOXL2 (0.64) HPGDLOXL2TSHRGAAALOX5
SCHEMBL2839532 0.82 LOXL2 (0.64) HPGDLOXL2TSHRGAAALOX5
SCHEMBL8323672 0.81 LOXL2 (0.58) HPGDLOXL2TSHRGAAALOX5
SCHEMBL21275558 0.81 LOXL2 (0.62) HPGDLOXL2TSHRGAAALOX5
SCHEMBL21318392 0.81 LOXL2 (0.62) HPGDLOXL2TSHRGAAALOX5
SCHEMBL20072395 0.81 LOXL2 (0.62) HPGDLOXL2TSHRGAAALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108395428-B Benzothiazole-triazole-isatin type compound and synthesis and application thereof 贵州医科大学 2021-02-02 CN claimed
CN-120961195-A Iron-loaded sulfonated carbon nitride heterogeneous catalyst and preparation method and application thereof 北京化工大学 2025-11-18 CN disclosed
CN-119119033-A Pyrazolopyridone compounds 百济神州有限公司 2024-12-13 CN disclosed
US-20240300951-A1 Pyrazolopyridinone Compounds BEIGENE LTD. (KY) 2024-09-12 US disclosed
US-20240270751-A1 Pyrazolopyridinone Compounds BEIGENE LTD. (KY) 2024-08-15 US disclosed
EP-4380936-A1 PYRAZOLOPYRIDINONE COMPOUNDS BeiGene, Ltd. (KY) 2024-06-12 EP disclosed
WO-2023011456-A1 PYRAZOLOPYRIDINONE COMPOUNDS BEIGENE, LTD. (KY) 2023-02-09 WO disclosed
CN-108395428-B Benzothiazole-triazole-isatin type compound and synthesis and application thereof 贵州医科大学 2021-02-02 CN disclosed
CN-108395428-B Benzothiazole-triazole-isatin type compound and synthesis and application thereof 贵州医科大学 2021-02-02 CN disclosed
US-9663508-B2 Biaryl acyl-sulfonamide compounds as sodium channel inhibitors AMGEN INC. (US) 2017-05-30 US disclosed
EP-1836158-A1 FUSED BICYCLIC CARBOXAMIDE DERIVATIVES FOR USE AS CXCR2 INHIBITORS IN THE TREATMENT OF INFLAMMATION Sanofi-Aventis Deutschland GmbH (DE) 2007-09-26 EP disclosed
WO-2006069656-A1 FUSED BICYCLIC CARBOXAMIDE DERIVATIVES FOR USE AS CXCR2 INHIBITORS IN THE TREATMENT OF INFLAMMATION SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-07-06 WO disclosed
EP-0795550-B1 Aniline derivatives having herbicidal activity their preparation and their use SANKYO CO (JP) 2002-06-05 EP disclosed
CN-1073097-C Aniline derivatives having herbicidal activity their prepn. and their use SANKYO CO (JP) 2001-10-17 CN disclosed
US-5736487-A HERBICIDES SANKYO COMPANY, LIMITED (JP) 1998-04-07 US disclosed
CN-1176962-A Aniline derivatives having herbicidal activity their prepn. and their use SANKYO CO (JP) 1998-03-25 CN disclosed
EP-0795550-A1 Aniline derivatives having herbicidal activity their preparation and their use SANKYO COMPANY LIMITED (JP) 1997-09-17 EP disclosed
EP-0222576-B1 HETEROCYCLIC OXOPHTHALAZINYL ACETIC ACIDS PFIZER INC. (US) 1992-03-18 EP disclosed
US-4939140-A ALDOSE REDUCTASE INHIBITORS PFIZER INC. (US) 1990-07-03 US disclosed
EP-0222576-A2 Heterocyclic oxophthalazinyl acetic acids PFIZER INC. (US) 1987-05-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240300951-A1 Pyrazolopyridinone Compounds NFATC1, CD4, PBK HPGD 1034/4885LOXL2 4062/4885TSHR 3432/4885
US-20240270751-A1 Pyrazolopyridinone Compounds NFATC1, CD4, PBK HPGD 1034/4885LOXL2 4062/4885TSHR 3432/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.