SCHEMBL486394

SCHEMBL486394

C=CN[C@H](CS)C(=O)O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3884487 1.00
SCHEMBL3884492 1.00
SCHEMBL15320712 0.83 FOLH1 (0.36)
SCHEMBL15320713 0.83 FOLH1 (0.36)
SCHEMBL19501717 0.80
SCHEMBL27529709 0.79
SCHEMBL4410363 0.79
SCHEMBL5088899 0.77 CA2 (0.41)
SCHEMBL8751952 0.77
SCHEMBL3669379 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3219325-B1 VARIANTS OF THE LANTIBIOTIC MU1140 AND OTHER LANTIBIOTICS WITH IMPROVED PHARMACOLOGICAL PROPERTIES AND STRUCTURAL FEATURES ORAGENICS INC (US) 2019-11-06 EP disclosed
US-9963488-B2 Variants of the lantibiotic MU1140 and other lantibiotics with improved pharmacological properties and structural features ORAGENICS, INC. (US) 2018-05-08 US disclosed
EP-3219325-A1 VARIANTS OF THE LANTIBIOTIC MU1140 AND OTHER LANTIBIOTICS WITH IMPROVED PHARMACOLOGICAL PROPERTIES AND STRUCTURAL FEATURES Oragenics, Inc. (US) 2017-09-20 EP disclosed
US-9120861-B2 Functional enhancement of antimicrobials MISSISSIPPI STATE UNIVERSITY (US) 2015-09-01 US disclosed
US-20150125503-A1 Variants of the Lantibiotic MU1140 and Other Lantibiotics with Improved Pharmacological Properties and Structural Features ORAGENICS, INC. 2015-05-07 US disclosed
EP-2833902-A1 VARIANTS OF THE LANTIBIOTIC MU1140 AND OTHER LANTIBIOTICS WITH IMPROVED PHARMACOLOGICAL PROPERTIES AND STRUCTURAL FEATURES Oragenics, Inc. (US) 2015-02-11 EP disclosed
WO-2013130349-A1 VARIANTS OF THE LANTIBIOTIC MU1140 AND OTHER LANTIBIOTICS WITH IMPROVED PHARMACOLOGICAL PROPERTIES AND STRUCTURAL FEATURES ORAGENICS, INC. (US) 2013-09-06 WO disclosed
EP-2411404-A1 DIFFERENTIALLY PROTECTED ORTHOGONAL LANTHIONINE TECHNOLOGY Oragenics, Inc. (US) 2012-02-01 EP disclosed
EP-1915389-B1 DIFFERENTIALLY PROTECTED ORTHOGONAL LANTHIONINE TECHNOLOGY ORAGENICS INC (US) 2011-06-08 EP disclosed
WO-2010117652-A1 DIFFERENTIALLY PROTECTED ORTHOGONAL LANTHIONINE TECHNOLOGY ORAGENICS, INC. (US) 2010-10-14 WO disclosed
US-20100145010-A1 Functional enhancement of antimicrobials MISSISSIPPI STATE UNIVERSITY 2010-06-10 US disclosed
US-20090215985-A1 DIFFERENTIALLY PROTECTED ORTHOGONAL LANTHIONINE TECHNOLOGY ORAGENICS, INC. 2009-08-27 US disclosed
US-7521529-B2 Differentially protected orthogonal lanthionine technology ORAGENICS, INC. (US) 2009-04-21 US disclosed
EP-1915389-A2 DIFFERENTIALLY PROTECTED ORTHOGONAL LANTHIONINE TECHNOLOGY Oragenics, Inc. (US) 2008-04-30 EP disclosed
WO-2007022012-A2 DIFFERENTIALLY PROTECTED ORTHOGONAL LANTHIONINE TECHNOLOGY ORAGENICS, INC. (US) 2007-02-22 WO disclosed
US-20070037963-A1 Lantibiotics; biosynthesis; solid phase synthesis; deblocking, deprotecting ORAGENICS, INC. 2007-02-15 US disclosed