SCHEMBL4864146

SCHEMBL4864146

C=CCOC(=S)C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.32
APP P05067 1/20 0.32
TSHR P16473 1/20 0.31
MAPT P10636 1/20 0.31
CACNA1B Q00975 1/20 0.31
APBA1 Q02410 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13351664 0.73 CYP3A4 (0.33) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL1082749 0.71 CYP3A4 (0.41) CYP3A4APPTSHRMAPTCACNA1B
SCHEMBL9286605 0.71 MAPT (0.36) CYP3A4TSHRMAPTCACNA1BAPBA1
SCHEMBL6695619 0.71 CYP3A4 (0.38) CYP3A4APPTSHRMAPTCACNA1B
SCHEMBL28427366 0.70 CYP3A4 (0.39) CYP3A4APPTSHRMAPTCACNA1B
SCHEMBL822080 0.70 CYP3A4 (0.31) CYP3A4
SCHEMBL29506833 0.70 CYP3A4 (0.39) CYP3A4APPTSHRMAPTCACNA1B
SCHEMBL11444238 0.70 CYP3A4 (0.39) CYP3A4APPTSHRMAPTCACNA1B
SCHEMBL31732818 0.70 CYP3A4 (0.31) CYP3A4
SCHEMBL28761387 0.70 CYP3A4 (0.39) CYP3A4APPTSHRMAPTCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470810-B2 Alkyl and aryl-thiotrifluoroacetates and process BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-30 US claimed
WO-2005073185-A1 NOVEL ALKYL- AND ARYL-THIOTRIFLUOROACETATES AND PROCESS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-08-11 WO claimed
US-20050159612-A1 Novel alkyl- and aryl-thiotrifluoroacetates and process BRISTOL-MYERS SQUIBB COMPANY 2005-07-21 US claimed
US-7470810-B2 Alkyl and aryl-thiotrifluoroacetates and process BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-30 US disclosed
WO-2005073185-A1 NOVEL ALKYL- AND ARYL-THIOTRIFLUOROACETATES AND PROCESS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-08-11 WO disclosed
US-20050159612-A1 Novel alkyl- and aryl-thiotrifluoroacetates and process BRISTOL-MYERS SQUIBB COMPANY 2005-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050159612-A1 Novel alkyl- and aryl-thiotrifluoroacetates and process TAF9, TAF1, TAF1L CYP3A4 3236/4885APP 2274/4885TSHR 126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.