SCHEMBL4865249

SCHEMBL4865249

Cc1cnc(C(Cc2ccccc2)NC(=O)OC(C)(C)C)[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR3 P32745 1/20 0.55
ALDH1A1 P00352 6/20 0.51
HPGD P15428 5/20 0.50
HTT P42858 5/20 0.50
NPSR1 Q6W5P4 5/20 0.50
LMNA P02545 4/20 0.50
TSHR P16473 3/20 0.50
PKM P14618 3/20 0.50
HSD17B10 Q99714 3/20 0.50
XBP1 P17861 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
ALOX15 P16050 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ATM Q13315 2/20 0.49
JAK2 O60674 3/20 0.48
PTPRB P23467 2/20 0.48
S1PR4 O95977 1/20 0.48
HSP90AA1 P07900 1/20 0.48
THRB P10828 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1197175 1.00 SSTR3 (0.55) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL22060193 0.88 SSTR3 (0.54) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL1197108 0.88 SSTR3 (0.54) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL20630809 0.86 SSTR3 (0.52) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL390451 0.86 SSTR3 (0.52) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL20630526 0.85 SSTR3 (0.52) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL1197182 0.81 ALDH1A1 (0.52) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL15875597 0.81 ALDH1A1 (0.52) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL1197116 0.80 ALDH1A1 (0.49) SSTR3ALDH1A1HPGDHTTNPSR1
SCHEMBL6791477 0.79 ALDH1A1 (0.58) ALDH1A1HPGDHTTNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981854-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS Brystol-Myers Squibb Company (US) 2008-10-22 EP disclosed
WO-2007070826-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-21 WO disclosed