SCHEMBL4867031

SCHEMBL4867031

CNCC1Cc2cc(Cl)cc(-c3ccc(F)c(Cl)c3)c2O1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.60
EZH2 Q15910 1/20 0.47
PRKAB2 O43741 1/20 0.38
PRKAG1 P54619 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAA1 Q13131 1/20 0.38
PRKAG3 Q9UGI9 1/20 0.38
PRKAG2 Q9UGJ0 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
HTR2A P28223 1/20 0.35
GRM2 Q14416 1/20 0.35
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
CHRM1 P11229 1/20 0.34
PTGS2 P35354 3/20 0.34
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
PTGS1 P23219 1/20 0.34
CYP11B1 P15538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4231239 0.92 AQP1 (0.58) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4218913 0.88 AQP1 (0.54) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4220623 0.88 AQP1 (0.54) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4231164 0.84 AQP1 (0.57) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL27707638 0.83 AQP1 (0.47) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4232174 0.82 AQP1 (0.67) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4230508 0.82 AQP1 (0.61) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4225480 0.81 AQP1 (0.65) AQP1EZH2PRKAB2PRKAG1PRKAA2
SCHEMBL4225947 0.81 AQP1 (0.67) AQP1EZH2HTR2ACHRM1SLC6A2
SCHEMBL27703101 0.81 AQP1 (0.53) AQP1EZH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101203216-A Dihydrobenzofuran derivatives and uses thereof WYETH CORP (US) 2008-06-18 CN disclosed
EP-1871355-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION Wyeth (US) 2008-01-02 EP disclosed
WO-2006116149-A1 NEW THERAPEUTIC COMBIANATIONS FOR THE TREATMENT OR PREVENTION OF DEPRESSION WYETH (US) 2006-11-02 WO disclosed