SCHEMBL4867443

SCHEMBL4867443

CCOC(=O)c1ccc(N2C(=O)[C@@H]3[C@@H]([C@@H]4C=C[C@H]3C4)S2(=O)=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.52
ATM Q13315 1/20 0.47
LMNA P02545 1/20 0.47
RAB9A P51151 1/20 0.46
TSHR P16473 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HPGD P15428 5/20 0.44
HTT P42858 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HSP90AA1 P07900 1/20 0.44
CACNA1B Q00975 1/20 0.44
APBA1 Q02410 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
KDM4E B2RXH2 2/20 0.42
MAPK1 P28482 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14254599 1.00 ALDH1A1 (0.52) ALDH1A1ATMLMNARAB9ATSHR
SCHEMBL5835332 0.82 CA1 (0.41) ALDH1A1SMN1; SMN2HPGDTDP1KDM4E
SCHEMBL5524587 0.80 ALDH1A1 (0.76) ALDH1A1ATMTSHRSMN1; SMN2HPGD
SCHEMBL14494335 0.73 ALDH1A1 (0.62) ALDH1A1ATMTSHRSMN1; SMN2HPGD
SCHEMBL5515220 0.71 SMN1; SMN2 (0.58) ALDH1A1ATMLMNATSHRSMN1; SMN2
SCHEMBL5524642 0.71 POLB (0.60) ALDH1A1ATMLMNATSHRSMN1; SMN2
SCHEMBL5835344 0.70 CA1 (0.41) ALDH1A1LMNASMN1; SMN2HPGDTDP1
SCHEMBL13483824 0.68 ALDH1A1 (0.58) ALDH1A1ATMTSHRSMN1; SMN2HPGD
SCHEMBL4705442 0.68 KAT2B (0.39) LMNATSHRSMN1; SMN2HTTNPSR1
SCHEMBL4705445 0.68 KAT2B (0.39) LMNATSHRSMN1; SMN2HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7342034-B2 Fused heterocyclic compounds and analogs thereof, modulators of nuclear hormone receptor function BRISTOL-MYERS SQUIBB COMPANY (US) 2008-03-11 US disclosed
US-7291637-B2 Fused heterocyclic compounds and analogs thereof, modulators of nuclear hormone receptor function BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-06 US disclosed