SCHEMBL4870538

SCHEMBL4870538

Cc1n[nH]c(C)c1-c1cnc2nc(N)nc(N3CCOCC3)c2n1.Nc1nc(N2CCOCC2)c2nc(-c3cnn(CC4OCCO4)c3)cnc2n1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.49
IKBKE Q14164 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
LRRK2 Q5S007 3/20 0.33
NUDT1 P36639 1/20 0.32
PIK3CA P42336 2/20 0.32
MTOR P42345 2/20 0.32
MET P08581 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
PIK3CD O00329 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4870532 0.90 NOS1 (0.37) NOS1IKBKETBK1LRRK2MET
SCHEMBL3765188 0.89 NOS1 (0.60) NOS1IKBKETBK1LRRK2PIK3CA
SCHEMBL3760468 0.84 NOS1 (0.60) NOS1LRRK2NUDT1PIK3CAMTOR
SCHEMBL3755618 0.77 NOS1 (0.62) NOS1LRRK2NUDT1PIK3CAPIK3CD
SCHEMBL3763426 0.76 NOS1 (0.61) NOS1LRRK2PIK3CAMTORPIM1
SCHEMBL3760285 0.74 NOS1 (0.59) NOS1LRRK2PIK3CAMTOR
SCHEMBL3765490 0.74 NOS1 (0.70) NOS1LRRK2PIK3CAPIM1PIK3CD
SCHEMBL3762264 0.73 NOS1 (0.71) NOS1PIK3CA
SCHEMBL3757137 0.72 IKBKE (0.46) NOS1IKBKETBK1MET
SCHEMBL3765592 0.70 NOS1 (0.64) NOS1NUDT1PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009079-A2 SUBSTITUTED PTERIDINES USEFUL FOR THE TREATMENT AND PREVENTION OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed