SCHEMBL4873041

SCHEMBL4873041

C[C@@H](O)[C@H](NC(=O)C1(CCNC(=O)OC(C)(C)C)C=CC(c2ccccc2)=CC1)C(=O)NO

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.38
CTSK P43235 3/20 0.38
AKT1 P31749 1/20 0.36
TSHR P16473 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
S1PR1 P21453 1/20 0.36
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
PSMB1 P20618 1/20 0.35
PSMB8 P28062 1/20 0.35
PSMB9 P28065 1/20 0.35
PSMB5 P28074 1/20 0.35
PSMB10 P40306 1/20 0.35
PSMB2 P49721 1/20 0.35
MMP13 P45452 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
APP P05067 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4873402 0.84 ANPEP (0.36) HDAC8
SCHEMBL5934160 0.83 CTSS (0.34) CTSSCTSKAKT1CTSLCTSB
SCHEMBL403598 0.82 ANPEP (0.35)
SCHEMBL4870451 0.76
SCHEMBL4873035 0.75 TSHR (0.35) CTSSCTSKTSHRMMP1MMP3
SCHEMBL404532 0.74 ANPEP (0.34)
SCHEMBL403350 0.73
SCHEMBL4236734 0.73
SCHEMBL4239586 0.73
SCHEMBL28745415 0.71 CTSS (0.42) CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7358359-B2 Antibacterial agents UNIVERSITY OF WASHINGTON (US) 2008-04-15 US disclosed