SCHEMBL4873605

SCHEMBL4873605

C[C@H](c1ncc[nH]1)c1cccc(F)c1F

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.58
ADRA2B P18089 2/20 0.58
ADRA2C P18825 2/20 0.58
F2RL1 P55085 15/20 0.46
TAAR1 Q96RJ0 1/20 0.41
PTGER3 P43115 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698055 1.00 ADRA2A (0.58) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL697224 0.88 ADRA2A (0.58) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL3532392 0.86 ADRA2A (0.57) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL13034019 0.86 ADRA2A (0.57) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL700615 0.86 ADRA2A (0.57) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL698140 0.82 ADRA2A (0.53) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL1573055 0.82 ADRA2A (0.51) ADRA2AADRA2BADRA2CF2RL1TAAR1
SCHEMBL714299 0.81 F2RL1 (0.59) F2RL1
SCHEMBL955822 0.81 F2RL1 (0.49) ADRA2AADRA2BADRA2CF2RL1
Demiditraz SCHEMBL696353 0.78 ADRA2A (0.61) ADRA2AADRA2BADRA2CF2RL1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981880-A2 USE OF 4-IMIDAZOLE DERIVATIVES FOR CNS DISORDERS F.HOFFMANN-LA ROCHE AG (CH) 2008-10-22 EP disclosed
WO-2007085556-A2 USE OF 4-IMIDAZOLE DERIVATIVES FOR CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-02 WO disclosed