SCHEMBL4874886

SCHEMBL4874886

O=c1oc2ccc(F)cc2cc1O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.61
CA1 P00915 2/20 0.61
CA2 P00918 2/20 0.61
CA9 Q16790 2/20 0.61
DAO P14920 3/20 0.59
HPGD P15428 2/20 0.59
TYR P14679 1/20 0.59
AKR1B1 P15121 1/20 0.59
NQO1 P15559 2/20 0.49
ATM Q13315 1/20 0.47
GPR35 Q9HC97 2/20 0.46
MAOA P21397 1/20 0.44
POLB P06746 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306505 0.81 CA12 (0.65) CA12CA1CA2CA9DAO
SCHEMBL1369097 0.79 ATM (0.58) CA12CA1CA2CA9ATM
SCHEMBL7803332 0.78 TYR (0.59) CA12CA1CA2CA9DAO
SCHEMBL11827623 0.78 MAOB (0.65) CA12CA1CA2CA9DAO
SCHEMBL11831412 0.78 CA12 (0.61) CA12CA1CA2CA9NQO1
SCHEMBL10602125 0.78 MAOB (0.68) CA12CA1CA2CA9NQO1
SCHEMBL9056428 0.78 CA12 (0.61) CA12CA1CA2CA9NQO1
SCHEMBL28994275 0.78 CA12 (0.57) CA12CA1CA2CA9NQO1
SCHEMBL21438975 0.78 GRIN1 (0.63) CA12CA1CA2CA9DAO
SCHEMBL11618896 0.77 CA12 (0.53) CA12CA1CA2CA9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080057529-A1 Method for Identifying Histone Deacetylase Inhibitors PALLAORO MICHELE 2008-03-06 US disclosed
EP-1697538-A1 METHOD FOR IDENTIFYING HISTONE DEACETYLASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2006-09-06 EP disclosed
WO-2005059167-A1 METHOD FOR IDENTIFYING HISTONE DEACETYLASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI SPA (IT) 2005-06-30 WO disclosed