SCHEMBL4875328

SCHEMBL4875328

N#Cc1cccc(C2CC2)c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.67
DRD3 P35462 11/20 0.67
CYP2D6 P10635 1/20 0.54
TSHR P16473 1/20 0.54
NFKB1 P19838 1/20 0.54
CASP1 P29466 1/20 0.54
NPSR1 Q6W5P4 1/20 0.52
USP30 Q70CQ3 1/20 0.46
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
ABCC9 O60706 1/20 0.44
ABCC8 Q09428 1/20 0.44
KCNJ11 Q14654 1/20 0.44
KCNJ8 Q15842 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28728225 0.93 DRD2 (0.59) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL31523251 0.92 DRD2 (0.73) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL14102178 0.91 DRD2 (0.58) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL13197442 0.91 DRD3 (0.58) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL28306714 0.91 DRD3 (0.58) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL4673932 0.91 DRD2 (0.58) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL13197443 0.91 DRD3 (0.58) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL2227921 0.90 DRD2 (0.71) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL4071635 0.89 DRD2 (0.59) DRD2DRD3CYP2D6TSHRNFKB1
SCHEMBL30809964 0.89 DRD2 (0.69) DRD2DRD3CYP2D6TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118390073-A Organic electrochemical synthesis method of cyclopropane compound 南京林业大学 2024-07-26 CN disclosed
CN-108289893-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2022-04-12 CN disclosed
CN-112341399-A 1,2, 4-triazole derivative compounds and application thereof in treating inflammatory bowel diseases 王健 2021-02-09 CN disclosed
CN-102753533-A Imidazolidinedione derivatives AUTIFONY THERAPEUTICS LTD 2012-10-24 CN disclosed
US-20080132477-A1 Macrocyclic Compounds Useful as Bace Inhibitors NOVARTIS AG (CH) 2008-06-05 US disclosed
CN-101103008-A Macrocyclic compounds useful as bace inhibitors NOVARTIS AG (CH) 2008-01-09 CN disclosed
EP-1851208-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS Novartis AG (CH) 2007-11-07 EP disclosed
WO-2006074950-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2006-07-20 WO disclosed
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP disclosed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP disclosed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132477-A1 Macrocyclic Compounds Useful as Bace Inhibitors BACE1, BACE2, APP DRD2 3124/4885DRD3 3013/4885CYP2D6 476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.