SCHEMBL4878360

SCHEMBL4878360

CNC1CCN(S(=O)(=O)c2cccc3c(O)nccc23)CC1.NC1CCN(S(=O)(=O)c2cccc3c(O)nccc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.43
ROCK1 Q13464 9/20 0.43
PRKX P51817 1/20 0.43
PRKCE Q02156 1/20 0.43
PRKCD Q05655 1/20 0.43
PRKD1 Q15139 1/20 0.43
ALOX5AP P20292 2/20 0.42
FEN1 P39748 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
EPHX2 P34913 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
COMT P21964 2/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
THPO P40225 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5086217 0.95 SMN1; SMN2 (0.46) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL5083072 0.91 ROCK2 (0.49) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL4728460 0.88 ALOX5AP (0.45) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL4728648 0.85 ROCK2 (0.45) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL5086408 0.81 CHRM1 (0.50) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL4728126 0.81 ROCK2 (0.43) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL4726171 0.81 CCR6 (0.47) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL4732315 0.78 MAPK1 (0.50) SMN1; SMN2EPHX2
SCHEMBL4725363 0.78 ROCK2 (0.48) ROCK2ROCK1PRKXPRKCEPRKCD
SCHEMBL2907238 0.77 POLB (0.56) ROCK2ROCK1PRKXPRKCEPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021210-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-02-21 WO disclosed