SCHEMBL4882526

SCHEMBL4882526

CN1CCN(c2ccc(-c3cnc4nc(N)nc(N5CCOCC5)c4n3)cn2)CC1.Cn1cc(-c2cnc3nc(N)nc(N4CCOCC4)c3n2)cn1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.58
ADK P55263 1/20 0.52
ATR Q13535 4/20 0.43
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
RET P07949 2/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
MET P08581 1/20 0.40
MTOR P42345 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3760382 0.94 NOS1 (0.66) NOS1ADKATRROCK2ROCK1
SCHEMBL3765490 0.88 NOS1 (0.70) NOS1ADK
SCHEMBL3756802 0.82 NOS1 (0.66) NOS1ADKATR
SCHEMBL3764506 0.81 NOS1 (0.63) NOS1ADKROCK2ROCK1
SCHEMBL3765371 0.79 NOS1 (0.75) NOS1ADKMTOR
SCHEMBL3761946 0.78 NOS1 (0.73) NOS1ADKMTOR
SCHEMBL3767213 0.78 NOS1 (0.64) NOS1ATRMTOR
SCHEMBL3763269 0.77 NOS1 (0.72) NOS1ADKATRMTOR
SCHEMBL3757061 0.77 NOS1 (0.72) NOS1ADKMTOR
SCHEMBL3765366 0.77 NOS1 (0.72) NOS1ADKATRMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009079-A2 SUBSTITUTED PTERIDINES USEFUL FOR THE TREATMENT AND PREVENTION OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed