SCHEMBL4883420

SCHEMBL4883420

CCCCCCCCCCCCCCOC(=O)CNC

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.64
EPHX1 P07099 1/20 0.60
FAAH O00519 2/20 0.58
RAD52 P43351 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
DGKA P23743 1/20 0.53
HTR2C P28335 1/20 0.51
ACHE P22303 6/20 0.48
TSHR P16473 2/20 0.48
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81047 1.00 NAAA (0.64) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL8377208 1.00 NAAA (0.64) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL7519633 1.00 NAAA (0.64) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL8379909 1.00 NAAA (0.64) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL5267200 1.00 NAAA (0.64) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL6566958 0.98 NAAA (0.62) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL394098 0.98 NAAA (0.62) NAAAEPHX1FAAHRAD52NPSR1
Hydrochloric Acid SCHEMBL5267197 0.98 NAAA (0.62) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL27285973 0.98 NAAA (0.62) NAAAEPHX1FAAHRAD52NPSR1
SCHEMBL168311 0.98 NAAA (0.61) NAAAEPHX1FAAHRAD52NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 153 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216036-B1 TRANSDERMAL ADMINISTRATION OF N-(2,5-DISUBSTITUTED PHENYL)-N'-(3-SUBSTITUTED PHENYL)-N'-METHYL GUANIDINES ALZA CORP (US) 2005-11-16 EP claimed
US-6960353-B2 Formulations for the transdermal administration of fenoldopam ALZA CORPORATION (US) 2005-11-01 US claimed
US-20040258742-A1 Transdermal administration of N-(2,5-disubstituted phenyl)-N'-(3-substituted phenyl)-N'-methyl guanidines VAN OSDOL WILLIAM WOODSON (US) 2004-12-23 US claimed
EP-1100476-B1 FORMULATIONS FOR THE TRANSDERMAL ADMINISTRATION OF FENOLDOPAM ALZA CORP (US) 2004-06-16 EP claimed
US-20040057987-A1 Novel formulations for the transdermal administration of fenoldopam VAN OSDOL WILLIAM W (US) 2004-03-25 US claimed
US-6699497-B1 PERMEATION ENHANCER ALZA CORPORATION 2004-03-02 US claimed
US-20030198662-A1 Transdermal administration of N-(2,5-disubstituted phenyl)-N'-(3-substituted phenyl)-N'-methyl guanidines VAN OSDOL WILLIAM WOODSON (US) 2003-10-23 US claimed
EP-1216036-A1 TRANSDERMAL ADMINISTRATION OF N-(2,5-DISUBSTITUTED PHENYL)-N'-(3-SUBSTITUTED PHENYL)-N'-METHYL GUANIDINES Alza Corporation (US) 2002-06-26 EP claimed
EP-1100476-A1 FORMULATIONS FOR THE TRANSDERMAL ADMINISTRATION OF FENOLDOPAM ALZA CORPORATION (US) 2001-05-23 EP claimed
WO-2001019352-A1 TRANSDERMAL ADMINISTRATION OF N-(2,5-DISUBSTITUTED PHENYL)-N'-(3-SUBSTITUTED PHENYL)-N'-METHYL GUANIDINES ALZA CORPORATION (US) 2001-03-22 WO claimed
WO-2000004886-A1 FORMULATIONS FOR THE TRANSDERMAL ADMINISTRATION OF FENOLDOPAM ALZA CORPORATION (US) 2000-02-03 WO claimed
EP-4736873-A1 ANTI-IL-4RALPHA ANTIBODY FORMULATION, PREPARATION METHOD THEREFOR, AND USE THEREOF Bio-Thera Solutions, Ltd. (CN) 2026-05-06 EP disclosed
US-20250257116-A1 ANTI-CLEAVAGE MUTANT OF CD16 FOR ENHANCING CELL FUNCTION NEUKIO BIOTHERAPEUTICS (SHANGHAI) CO., LTD. (CN) 2025-08-14 US disclosed
CN-119968452-A Perfume mixture (VI) 西姆莱斯股份公司 2025-05-09 CN disclosed
US-20250134934-A1 IMPROVED METHODS FOR DECELLULARIZING EXTRACELLULAR MATRIX (ECM) AND PREPARING DECELLULARIZED ECM GELS AND USES THEREOF REGENX SCIENCE, INC. (US) 2025-05-01 US disclosed
EP-1169025-A2 TRANSDERMAL DRUG DELIVERY DEVICES COMPRISING A POLYURETHANE DRUG RESERVOIR Alza Corporation (US) 2002-01-09 EP disclosed
EP-1100476-A1 FORMULATIONS FOR THE TRANSDERMAL ADMINISTRATION OF FENOLDOPAM ALZA CORPORATION (US) 2001-05-23 EP disclosed
WO-2001019352-A1 TRANSDERMAL ADMINISTRATION OF N-(2,5-DISUBSTITUTED PHENYL)-N'-(3-SUBSTITUTED PHENYL)-N'-METHYL GUANIDINES ALZA CORPORATION (US) 2001-03-22 WO disclosed
WO-2000059483-A2 TRANSDERMAL DRUG DELIVERY DEVICES COMPRISING A POLYURETHANE DRUG RESERVOIR ALZA CORPORATION (US) 2000-10-12 WO disclosed
WO-2000004886-A1 FORMULATIONS FOR THE TRANSDERMAL ADMINISTRATION OF FENOLDOPAM ALZA CORPORATION (US) 2000-02-03 WO disclosed