SCHEMBL488876

SCHEMBL488876

CC1(C)OB(c2ccc(NS(=O)(=O)CCN3CCC(O)CC3)cc2)OC1(C)C

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 13/20 0.49
CA2 P00918 13/20 0.49
CA9 Q16790 13/20 0.49
CA12 O43570 1/20 0.49
CA3 P07451 1/20 0.49
CA4 P22748 1/20 0.49
CA6 P23280 1/20 0.49
CA5A P35218 1/20 0.49
CA7 P43166 1/20 0.49
CA14 Q9ULX7 1/20 0.49
CA5B Q9Y2D0 1/20 0.49
KDM1A O60341 1/20 0.41
TERT O14746 2/20 0.36
CYP2D6 P10635 1/20 0.36
OPRK1 P41145 1/20 0.36
PARP1 P09874 1/20 0.35
JAK2 O60674 1/20 0.34
JAK3 P52333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488842 0.94 CA1 (0.47) CA1CA2CA9CA12CA3
SCHEMBL488765 0.88 KDM1A (0.40) CA1CA2CA9CA12CA3
SCHEMBL488897 0.88 CA1 (0.54) CA1CA2CA9CA12CA3
SCHEMBL1601710 0.86 CA1 (0.53) CA1CA2CA9CA12CA3
SCHEMBL488908 0.86 CA1 (0.53) CA1CA2CA9CA12CA3
SCHEMBL488839 0.85 CA1 (0.52) CA1CA2CA9CA12CA3
SCHEMBL488793 0.84 CA1 (0.48) CA1CA2CA9CA12CA3
SCHEMBL488906 0.82 CA1 (0.46) CA1CA2CA9CA12CA3
SCHEMBL488764 0.82 CYP2D6 (0.38) CA1CA2CA9CA12CA3
SCHEMBL488959 0.80 CA1 (0.46) CA1CA2CA9CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed