SCHEMBL488765

SCHEMBL488765

CC1(C)OB(c2cccc(NS(=O)(=O)CCN3CCC(O)CC3)c2)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.40
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
SRC P12931 2/20 0.36
CA12 O43570 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
TERT O14746 1/20 0.34
DRD2 P14416 1/20 0.34
LPL P06858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
CYP2D6 P10635 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL488764 0.94 CYP2D6 (0.38) KDM1ACA1CA2CA9SRC
SCHEMBL488274 0.89 SRC (0.44) KDM1ACA1CA2CA9SRC
SCHEMBL488893 0.88 SRC (0.44) KDM1ACA1CA2CA9SRC
SCHEMBL488876 0.88 CA1 (0.49) KDM1ACA1CA2CA9CA12
SCHEMBL488233 0.87 MEN1 (0.40) CA1CA2CA9SRCCA12
SCHEMBL488629 0.85 SMN1; SMN2 (0.38) KDM1ACA1CA2CA9SRC
SCHEMBL488672 0.83 ROCK1 (0.36) KDM1ACA1CA2CA9SRC
SCHEMBL488842 0.82 CA1 (0.47) KDM1ACA1CA2CA9CA12
SCHEMBL488724 0.82 PARP1 (0.37) CA1CA2CA9CA12CA3
SCHEMBL488841 0.78 CA1 (0.38) CA1CA2CA9CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed