SCHEMBL4894685

SCHEMBL4894685

Nc1ccccc1C(NC(=O)CCc1ccccc1)C(=O)Nc1ccc(Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.56
KMT2A Q03164 3/20 0.56
HTT P42858 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
RAB9A P51151 2/20 0.47
MEN1 O00255 2/20 0.45
CNR1 P21554 2/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
NPC1 O15118 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
UTS2R Q9UKP6 1/20 0.45
SLC6A9 P48067 1/20 0.45
SLC6A5 Q9Y345 1/20 0.45
RORC P51449 1/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2684787 0.81 HDAC1 (0.56) MAPTKMT2AHTTNPSR1MEN1
SCHEMBL2685332 0.78 HDAC1 (0.49) MAPTKMT2AHTTNPSR1HDAC1
SCHEMBL3678030 0.76 MAPT (0.77) MAPTKMT2AHTTNPSR1RAB9A
SCHEMBL2687809 0.71 HDAC1 (0.56) KMT2AMEN1HDAC1HDAC6RORC
SCHEMBL5902414 0.71 MAPT (0.77) MAPTKMT2AHTTRAB9AMEN1
SCHEMBL2686100 0.70 HDAC1 (0.58) KMT2AMEN1HDAC1HDAC6ALDH1A1
SCHEMBL2684625 0.70 HDAC1 (0.59) HDAC1HDAC6RORC
SCHEMBL2356413 0.70 HDAC1 (0.72) MAPTKMT2AHTTRAB9AMEN1
SCHEMBL15350108 0.69 HDAC1 (0.73) MAPTKMT2AHTTRAB9AMEN1
SCHEMBL10198474 0.68 MAPT (0.77) MAPTKMT2AHTTRAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-A2 INHIBITORS OF HISTONE DEACETYLASE Merck & Co., Inc. (US) 2008-11-19 EP disclosed
WO-2007100657-A2 INHIBITORS OF HISTONE DEACETYLASE MERCK & CO., INC. (US) 2007-09-07 WO disclosed