SCHEMBL4897323

SCHEMBL4897323

NS(=O)(=O)c1ccc(CNc2c(Nc3ccc4[nH]cnc4c3)c(=O)c2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.48
ROCK1 Q13464 4/20 0.48
CLK4 Q9HAZ1 4/20 0.48
NEK4 P51957 3/20 0.48
PKN2 Q16513 3/20 0.48
AURKB Q96GD4 3/20 0.48
ROCK2 O75116 2/20 0.48
MAP4K4 O95819 2/20 0.48
PRKG2 Q13237 2/20 0.48
EEF2K O00418 1/20 0.48
CLK2 P49760 1/20 0.48
PRKX P51817 1/20 0.48
TAOK1 Q7L7X3 1/20 0.48
PBK Q96KB5 1/20 0.48
SLK Q9H2G2 1/20 0.48
MAP3K20 Q9NYL2 1/20 0.48
CA1 P00915 12/20 0.45
CA2 P00918 12/20 0.45
CA7 P43166 1/20 0.45
CA13 Q8N1Q1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4905370 0.90 ROCK1 (0.46) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4598765 0.89 ROCK2 (0.43) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4908463 0.88 ROCK1 (0.45) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4910893 0.87 ROCK1 (0.47) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4908343 0.85 ROCK1 (0.46) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4598260 0.85 ROCK1 (0.47) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL14066718 0.85 MAPKAPK2 (0.54) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4908067 0.83 GSK3B (0.44) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4908588 0.83 QPCT (0.48) GSK3BROCK1CLK4NEK4PKN2
SCHEMBL4904962 0.82 GSK3B (0.47) GSK3BROCK1CLK4NEK4PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080234266-A1 Squaric Acid Derivatives II MERCK PATENT GESELLSCHAFT (DE) 2008-09-25 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234266-A1 Squaric Acid Derivatives II CHEK2, CHEK1, SGK3 GSK3B 132/4885ROCK1 713/4885CLK4 133/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.