SCHEMBL4901986

SCHEMBL4901986

O=C(NNC(=S)N[C@H](Cc1cccnc1)CN1C(=O)c2ccccc2C1=O)c1ccc2cnccc2c1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 3/20 0.40
GAA P10253 2/20 0.40
AKT1 P31749 2/20 0.40
PKM P14618 1/20 0.39
DRD4 P21917 1/20 0.39
CDK2 P24941 1/20 0.39
DRD2 P14416 2/20 0.38
DRD3 P35462 1/20 0.38
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903498 1.00 ALDH1A1 (0.42) ALDH1A1KDM4EPOLBGAAAKT1
SCHEMBL4891405 0.95 AKT1 (0.41) ALDH1A1GAAAKT1CDK2NAMPT
SCHEMBL4896077 0.95 AKT1 (0.41) ALDH1A1GAAAKT1CDK2NAMPT
SCHEMBL4781246 0.95 AKT1 (0.41) ALDH1A1GAAAKT1CDK2NAMPT
SCHEMBL4899142 0.93 AKT1 (0.41) ALDH1A1AKT1CDK2NAMPT
SCHEMBL4900162 0.93 AKT1 (0.41) ALDH1A1AKT1CDK2NAMPT
SCHEMBL4898951 0.90 AKT1 (0.41) ALDH1A1KDM4EAKT1
SCHEMBL4899055 0.90 GAA (0.41) ALDH1A1KDM4EGAAAKT1
SCHEMBL4904361 0.90 AKT1 (0.41) ALDH1A1KDM4EPOLBGAAAKT1
SCHEMBL4901998 0.90 AKT1 (0.41) ALDH1A1KDM4EPOLBGAAAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith D SIDOCKY NEIL R 2008-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith JAK2, CHEK2, MTOR ALDH1A1 1752/4885KDM4E 1212/4885POLB 2428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.