SCHEMBL4902455

SCHEMBL4902455

COC(=O)c1ccc(-c2cncc[n+]2[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
SLC2A1 P11166 1/20 0.45
CYP19A1 P11511 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
KDM4E B2RXH2 2/20 0.44
GAA P10253 2/20 0.44
MAPT P10636 2/20 0.44
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA12 O43570 3/20 0.43
CA9 Q16790 3/20 0.43
CA14 Q9ULX7 3/20 0.43
SETD7 Q8WTS6 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA7 P43166 1/20 0.41
HTT P42858 1/20 0.40
MAPK1 P28482 1/20 0.40
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4907831 0.78 ALDH1A1 (0.46) ALDH1A1SLC2A1CYP19A1CYP11B1CYP11B2
SCHEMBL14164169 0.78 TSHR (0.50) ALDH1A1KDM4EMAPTCA1CA2
SCHEMBL16369789 0.73 ALDH1A1 (0.43) ALDH1A1CYP19A1CYP11B1CYP11B2KDM4E
SCHEMBL14164179 0.72 TDP1 (0.59) ALDH1A1SLC2A1CYP19A1CYP11B1CYP11B2
SCHEMBL743734 0.72 CA1 (0.57) ALDH1A1KDM4EMAPTCA1CA2
SCHEMBL741537 0.71 HDAC1 (0.58) ALDH1A1KDM4ECA1CA2CA12
SCHEMBL13019478 0.71 HDAC1 (0.58) ALDH1A1KDM4ECA1CA2CA12
SCHEMBL2345607 0.71 CYP19A1 (0.74) ALDH1A1SLC2A1CYP19A1CYP11B1CYP11B2
SCHEMBL30109243 0.70 ALDH1A1 (0.56) ALDH1A1SLC2A1CYP19A1CYP11B1CYP11B2
SCHEMBL14886472 0.70 ALDH1A1 (0.56) ALDH1A1SLC2A1CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080132698-A1 Use of N-oxide compounds in coupling reactions UNIVERSITY OF OTTAWA 2008-06-05 US disclosed
US-20080132698-A1 Use of N-oxide compounds in coupling reactions UNIVERSITY OF OTTAWA 2008-06-05 US disclosed
US-20080132698-A1 Use of N-oxide compounds in coupling reactions UNIVERSITY OF OTTAWA 2008-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132698-A1 Use of N-oxide compounds in coupling reactions CYP4X1, CYP4F3, CYP1A2 ALDH1A1 1518/4885SLC2A1 3053/4885CYP19A1 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.