SCHEMBL4903437

SCHEMBL4903437

Cc1ccc(C(=O)Nc2ccc(C)c(Nc3nccc(-c4ccccn4)n3)c2)cc1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 12/20 0.73
ABL1 P00519 12/20 0.73
BCR P11274 7/20 0.73
PDGFRB P09619 5/20 0.73
EGFR P00533 1/20 0.68
PRKCA P17252 1/20 0.68
KIT P10721 6/20 0.60
ABL2 P42684 2/20 0.59
KDR P35968 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4899586 0.92 PDGFRA (0.74) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4901380 0.92 PDGFRA (0.66) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4902233 0.91 PDGFRA (0.64) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4903235 0.90 PDGFRA (0.63) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4899582 0.90 ABL1 (0.75) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4904973 0.88 PDGFRA (0.78) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4903298 0.87 ABL1 (0.59) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4899247 0.87 ABL1 (0.73) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4905315 0.87 PDGFRA (0.61) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL4897577 0.85 ABL1 (0.60) PDGFRAABL1BCRPDGFRBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080187575-A1 Pyrimidine Derivatives VICHEM CHEMIE KFT (HU) 2008-08-07 US claimed
EP-1786781-A2 PYRIMIDINE DERIVATIVES GPC Biotech AG (DE) 2007-05-23 EP claimed
WO-2006021458-A2 PYRIMIDINE DERIVATIVES GPC BIOTECH AG (DE) 2006-03-02 WO claimed
US-20080187575-A1 Pyrimidine Derivatives VICHEM CHEMIE KFT (HU) 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080187575-A1 Pyrimidine Derivatives TYMP, TDP1, PNP PDGFRA 373/4885ABL1 2843/4885BCR 2315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.