SCHEMBL4903540

SCHEMBL4903540

CCn1c(N(C)C(=O)O)c(C(=O)Nc2ccc(Oc3ccnc4cc(OC)ccc34)c(F)c2)c(=O)n1-c1ccccc1

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.81
KDR P35968 20/20 0.81
IGF1R P08069 19/20 0.81
MST1R Q04912 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2354420 0.92 MET (0.81) METKDRIGF1R
SCHEMBL783420 0.90 MET (1.00) METKDRIGF1RMST1R
SCHEMBL4903552 0.86 MET (0.83) METKDRIGF1RMST1R
SCHEMBL198584 0.85 MET (1.00) METKDRIGF1RMST1R
SCHEMBL198400 0.85 MET (1.00) METKDRIGF1RMST1R
SCHEMBL201049 0.84 MET (0.87) METKDRIGF1RMST1R
SCHEMBL199470 0.84 MET (0.87) METKDRIGF1RMST1R
SCHEMBL200685 0.84 MET (0.91) METKDRIGF1RMST1R
SCHEMBL197413 0.84 MET (1.00) METKDRIGF1RMST1R
SCHEMBL198809 0.84 MET (1.00) METKDRIGF1RMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881976-A1 SUBSTITUTED AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS Amgen Inc., (US) 2008-01-30 EP claimed
WO-2006116713-A1 SUBSTITUTED AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS AMGEN INC. (US) 2006-11-02 WO claimed