SCHEMBL4905069

SCHEMBL4905069

C[C@@H](Nc1c(N(c2nc3ccccc3[nH]2)C(F)(F)F)c(=O)c1=O)c1cccc(O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 4/20 0.44
NLRP3 Q96P20 1/20 0.36
TEAD4 Q15561 1/20 0.35
COASY Q13057 1/20 0.34
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CXCR2 P25025 2/20 0.33
CXCR1 P25024 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 3/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4908560 1.00 MAPKAPK2 (0.44) MAPKAPK2NLRP3TEAD4COASYNPC1
SCHEMBL4915780 0.63 MAPKAPK2 (0.54) MAPKAPK2NLRP3HTTRAB9ASMN1; SMN2
SCHEMBL4927735 0.63 MAPKAPK2 (0.54) MAPKAPK2NLRP3HTTRAB9ASMN1; SMN2
SCHEMBL4366319 0.62 MAPKAPK2 (1.00) MAPKAPK2MAPK1CYP2D6
SCHEMBL1228404 0.61 MAPKAPK2 (0.61) MAPKAPK2MAPK1CYP2D6KDR
SCHEMBL4598811 0.61 MAPKAPK2 (0.61) MAPKAPK2MAPK1CYP2D6
SCHEMBL4596962 0.61 MAPKAPK2 (0.61) MAPKAPK2MAPK1CYP2D6
SCHEMBL4928754 0.60 MAPKAPK2 (0.56) MAPKAPK2MAPK1CYP2D6
SCHEMBL4916066 0.60 MAPKAPK2 (0.63) MAPKAPK2NLRP3MAPK1CYP2D6
SCHEMBL4914736 0.59 MAPKAPK2 (0.70) MAPKAPK2CXCR2CXCR1MAPK1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080234266-A1 Squaric Acid Derivatives II MERCK PATENT GESELLSCHAFT (DE) 2008-09-25 US claimed
US-20080234266-A1 Squaric Acid Derivatives II MERCK PATENT GESELLSCHAFT (DE) 2008-09-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234266-A1 Squaric Acid Derivatives II CHEK2, CHEK1, SGK3 MAPKAPK2 346/4885NLRP3 3953/4885TEAD4 2520/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.