SCHEMBL4906104

SCHEMBL4906104

CCc1ccc(S(=O)(=O)NCCc2nc(-c3ccc(F)cc3)sc2C)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 0.45
MAPT P10636 6/20 0.45
THRB P10828 2/20 0.44
LMNA P02545 3/20 0.43
POLB P06746 3/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
METAP2 P50579 2/20 0.40
TAAR1 Q96RJ0 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4906600 0.93 MAPT (0.46) TP53MAPTTHRBLMNAPPARG
SCHEMBL4911992 0.91 MAPT (0.48) TP53MAPTTHRBLMNAPOLB
SCHEMBL4904471 0.91 MAPT (0.46) TP53MAPTTHRBLMNAPPARG
SCHEMBL4904282 0.91 LMNA (0.48) TP53MAPTTHRBLMNAPOLB
SCHEMBL4899406 0.90 MAPT (0.45) TP53MAPTTHRBLMNAPOLB
SCHEMBL4906394 0.89 LMNA (0.41) TP53MAPTTHRBLMNAPOLB
SCHEMBL4905611 0.89 MAPT (0.42) TP53MAPTLMNA
SCHEMBL4899205 0.89 PPARA (0.48) TP53MAPTTHRBLMNAPPARG
SCHEMBL4905792 0.88 TP53 (0.44) TP53MAPTTHRBLMNAPOLB
SCHEMBL4906613 0.86 MAPT (0.44) TP53MAPTTHRBLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20050288340-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PFIZER INC 2005-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288340-A1 Substituted heteroaryl- and phenylsulfamoyl compounds PPARA, PPARG, PPARD TP53 3421/4885MAPT 1786/4885THRB 160/4885
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PPARA, PPARG, PPARD TP53 3421/4885MAPT 1786/4885THRB 160/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.