SCHEMBL4907283

SCHEMBL4907283

CCN(c1csc(-c2ccc(C)cc2)n1)S(=O)(=O)c1cc(C)c(C)c(C(=O)OC)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.42
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 3/20 0.37
TSHR P16473 2/20 0.37
MAPT P10636 4/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4902485 0.93 TP53 (0.40) TP53NPC1RAB9AALDH1A1TSHR
SCHEMBL4900904 0.91 NR1I2 (0.36) TP53NPC1RAB9AALDH1A1TSHR
SCHEMBL4902470 0.90 TP53 (0.43) TP53NPC1POLBRAB9AALDH1A1
SCHEMBL4906743 0.89 ALDH1A1 (0.44) TP53NPC1POLBRAB9AALDH1A1
SCHEMBL4898066 0.87 ALDH1A1 (0.39) TP53POLBALDH1A1TSHRMAPT
SCHEMBL4897618 0.87 TP53 (0.42) TP53NPC1POLBRAB9AALDH1A1
SCHEMBL4899693 0.84 TP53 (0.40) TP53NPC1RAB9AALDH1A1TSHR
SCHEMBL4904959 0.84 MAPT (0.39) TP53NPC1RAB9AALDH1A1TSHR
SCHEMBL4904147 0.82 ALDH1A1 (0.45) TP53NPC1RAB9AALDH1A1TSHR
SCHEMBL4902584 0.82 MAPT (0.43) TP53NPC1RAB9AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20060229363-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds HAMANAKA ERNEST S 2006-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229363-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds PPARA, PPARG, PPARD TP53 3260/4885NPC1 50/4885POLB 1488/4885
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PPARA, PPARG, PPARD TP53 3421/4885NPC1 59/4885POLB 1807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.