SCHEMBL4909397

SCHEMBL4909397

N[C@H]1CCN(c2ccc(I)cn2)C1.O=C(O)N[C@H]1CCN(c2ccc(I)cn2)C1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA12 O43570 20/20 0.47
CA1 P00915 20/20 0.47
CA2 P00918 20/20 0.47
CA4 P22748 20/20 0.47
CA7 P43166 20/20 0.47
CA9 Q16790 20/20 0.47
TRPV1 Q8NER1 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780968 0.93 CA12 (0.49) CA12CA1CA2CA4CA7
SCHEMBL14196276 0.84 HRH4 (0.46)
SCHEMBL14223014 0.84 HRH4 (0.46)
SCHEMBL14222473 0.84 HRH4 (0.46)
Hydrochloric Acid SCHEMBL4795755 0.83 HRH4 (0.45)
SCHEMBL1749349 0.82 CA12 (0.53) CA12CA1CA2CA4CA7
SCHEMBL14196277 0.80 PDE10A (0.48) CA12CA1CA2CA4CA7
SCHEMBL4885872 0.79 HRH4 (0.49) CA12CA1CA2CA4CA7
SCHEMBL15205294 0.78 TRPV1 (0.50) CA12CA1CA2CA4CA7
SCHEMBL997974 0.78 TRPV1 (0.50) CA12CA1CA2CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008041090-A1 MALANIN CONCENTRATING HORMONE RECEPTOR-1 ANTAGONIST PYRIDINONES PFIZER LIMITED (GB) 2008-04-10 WO disclosed