SCHEMBL4933296

SCHEMBL4933296

CN1CCC(Oc2cccc(CNC(=O)c3cccc(Oc4ccccc4)c3)c2)CC1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC5A7 Q9GZV3 3/20 0.60
KMT2A Q03164 4/20 0.57
MEN1 O00255 3/20 0.57
CHRM3 P20309 1/20 0.55
PABPC1 P11940 1/20 0.52
NPC1 O15118 3/20 0.52
APOBEC3A P31941 1/20 0.52
APOBEC3G Q9HC16 1/20 0.52
MMP13 P45452 1/20 0.51
OPRK1 P41145 1/20 0.51
FFAR1 O14842 1/20 0.51
MAOA P21397 1/20 0.50
ROCK2 O75116 1/20 0.49
CCR3 P51677 1/20 0.49
POLB P06746 1/20 0.49
MAPK14 Q16539 1/20 0.49
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4930039 0.93 MAPK14 (0.58) SLC5A7KMT2AMEN1MMP13FFAR1
SCHEMBL4666647 0.87 SLC5A7 (0.54) SLC5A7KMT2AMEN1NPC1MAOA
SCHEMBL4934208 0.87 SLC5A7 (0.54) SLC5A7KMT2AMEN1NPC1APOBEC3A
SCHEMBL14026963 0.87 LMNA (0.64) SLC5A7KMT2AMEN1PABPC1NPC1
Hydrochloric Acid SCHEMBL4666207 0.86 LMNA (0.63) SLC5A7KMT2AMEN1PABPC1NPC1
SCHEMBL22130619 0.86 SLC5A7 (0.55) SLC5A7KMT2AMEN1PABPC1NPC1
SCHEMBL4933614 0.84 LMNA (0.53) SLC5A7KMT2AMEN1
SCHEMBL14026961 0.84 SLC5A7 (0.54) SLC5A7KMT2AMEN1NPC1APOBEC3A
SCHEMBL4932164 0.83 SLC5A7 (0.68) SLC5A7KMT2AMEN1NPC1MMP13
SCHEMBL4933009 0.83 SLC5A7 (0.57) SLC5A7KMT2AMEN1MMP13FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080269275-A1 Novel Mchr1 Antagonists and Their Use for the Treatment of Mchr1 Mediated Conditions and Disorders ASTRAZENECA AB (SE) 2008-10-30 US claimed
US-20080269275-A1 Novel Mchr1 Antagonists and Their Use for the Treatment of Mchr1 Mediated Conditions and Disorders ASTRAZENECA AB (SE) 2008-10-30 US disclosed
US-20080269275-A1 Novel Mchr1 Antagonists and Their Use for the Treatment of Mchr1 Mediated Conditions and Disorders ASTRAZENECA AB (SE) 2008-10-30 US disclosed
US-20080269275-A1 Novel Mchr1 Antagonists and Their Use for the Treatment of Mchr1 Mediated Conditions and Disorders ASTRAZENECA AB (SE) 2008-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080269275-A1 Novel Mchr1 Antagonists and Their Use for the Treatment of Mchr1 Mediated Conditions and Disorders MCHR1, MCHR2, HCRTR1 SLC5A7 854/4885KMT2A 704/4885MEN1 501/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.