SCHEMBL4936099

SCHEMBL4936099

CCCC(Br)C(=O)c1ccc(I)cc1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.58
SLC6A3 Q01959 10/20 0.55
SLC6A2 P23975 8/20 0.55
SLC6A4 P31645 5/20 0.55
TPMT P51580 1/20 0.41
FOLH1 Q04609 3/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
PDPK1 O15530 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4935111 0.84 SLC6A3 (0.56) GSK3BSLC6A3SLC6A2SLC6A4CA1
SCHEMBL4937398 0.84 SLC6A3 (0.54) GSK3BSLC6A3SLC6A2SLC6A4
SCHEMBL17644172 0.84 SLC6A2 (0.54) SLC6A3SLC6A2SLC6A4CA1CA2
SCHEMBL4936186 0.82 SLC6A3 (0.55) SLC6A3SLC6A2SLC6A4CA1CA2
SCHEMBL2823791 0.81 SLC6A2 (0.53) GSK3BSLC6A3SLC6A2
SCHEMBL4935875 0.81 SLC6A2 (0.53) GSK3BSLC6A3SLC6A2
SCHEMBL4936027 0.81 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4
SCHEMBL4932919 0.79 SLC6A2 (0.57) GSK3BSLC6A3SLC6A2SLC6A4CA1
SCHEMBL4936697 0.79 SLC6A2 (0.57) SLC6A3SLC6A2SLC6A4CA1CA2
SCHEMBL4929359 0.78 GSK3B (0.62) GSK3BSLC6A3SLC6A2SLC6A4CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080234498-A1 Pyrovalerone Analogues and Therapeutic Uses Thereof PRESIDENT AND FELLOW OF HARVARD COLLEGE (US) 2008-09-25 US disclosed
EP-1670755-A4 PYROVALERONE ANALOGS AND THERAPEUTIC USES THEREOF HARVARD COLLEGE (US) 2007-02-28 EP disclosed
EP-1670755-A2 PYROVALERONE ANALOGS AND THERAPEUTIC USES THEREOF President And Fellows of Harvard College (US) 2006-06-21 EP disclosed
WO-2005034878-A2 PYROVALERONE ANALOGS AND THERAPEUTIC USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2005-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234498-A1 Pyrovalerone Analogues and Therapeutic Uses Thereof SLC6A2, SLC6A4, SLC6A3 GSK3B 539/4885SLC6A3 3/4885SLC6A2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.