SCHEMBL4936749

SCHEMBL4936749

CCC=C[CH]C=CCCC

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.41
PPARA Q07869 1/20 0.34
TSHR P16473 2/20 0.32
ALDH1A1 P00352 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28756777 0.91 TSHR (0.37) TSHRALDH1A1
SCHEMBL6474026 0.88
SCHEMBL732789 0.88
SCHEMBL732788 0.88
SCHEMBL6474469 0.88
SCHEMBL6480047 0.88
SCHEMBL15195021 0.85 TRPA1 (0.43) TRPA1PPARATSHRALDH1A1
SCHEMBL15195019 0.85 TRPA1 (0.43) TRPA1PPARATSHRALDH1A1
SCHEMBL28767917 0.85 TRPA1 (0.43) TRPA1PPARATSHRALDH1A1
SCHEMBL17504426 0.83 TSHR (0.43) TRPA1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024133845-A1 CONJUGATES COMPRISING A PHOSPHORUS(V) MOIETY AND A DRUG TUBULIS GMBH (DE) 2024-06-27 WO disclosed
CN-117736207-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-03-22 CN disclosed
US-11690282-B2 Organic solar cell LG CHEM, LTD. (KR) 2023-06-27 US disclosed
WO-2023106175-A1 URACIL COMPOUND, GERMICIDE FOR AGRICULTURAL AND HORTICULTURAL USE, NEMATICIDE, AND ANTIFUNGAL AGENT FOR MEDICAL AND ANIMAL USE 日本曹達株式会社 2023-06-15 WO disclosed
WO-2023053082-A1 LECTIN-DRUG CONJUGATES UNICHEM LABORATORIES LIMITED (IN) 2023-04-06 WO disclosed
WO-2023017699-A1 3-SUBSTITUTED URACIL COMPOUND, AGRICULTURAL AND HORTICULTURAL GERMICIDE, NEMATICIDE, AND MEDICAL AND ANIMAL ANTIFUNGAL AGENT 日本曹達株式会社 2023-02-16 WO disclosed
WO-2023276813-A1 PYRIDAZINONE COMPOUND, AGRICULTURAL AND HORTICULTURAL GERMICIDE, NEMATICIDE, AND MEDICAL AND ANIMAL ANTIFUNGAL AGENT 日本曹達株式会社 2023-01-05 WO disclosed
CN-107949645-B Use of hydrophobically associating copolymers as binders for granulation of metal-containing ores 巴斯夫欧洲公司 2021-03-12 CN disclosed
CN-108336239-B Organic light emitting element 株式会社LG化学 2020-06-23 CN disclosed
CN-105567717-B It is incorporated into the antibody drug conjugates (ADC) of 191P4D12 albumen Algens Co.,Ltd. (US) 2019-10-29 CN disclosed
EP-1844051-A1 THIENOPYRROLES USEFUL IN THE TREATMENT OF INFLAMMATION Biolipox AB (SE) 2007-10-17 EP disclosed
WO-2007109633-A2 ORGANOTELLURIUM AND SELENIUM-BASED ANTIMICROBIAL ANTIMICROBIAL FORMULATIONS AND ARTICLES ANDOVER HEALTHCARE, INC. (US) 2007-09-27 WO disclosed
EP-1817336-A2 AURISTATINS HAVING AN AMINOBENZOIC ACID UNIT AT THE N TERMINUS Seattle Genetics, Inc. (US) 2007-08-15 EP disclosed
WO-2006132670-A2 AURISTATINS HAVING AN AMINOBENZOIC ACID UNIT AT THE N TERMINUS SEATTLE GENETICS, INC. (US) 2006-12-14 WO disclosed
WO-2006077412-A1 THIENOPYRROLES USEFUL IN THE TREATMENT OF INFLAMMATION BIOLIPOX AB (SE) 2006-07-27 WO disclosed
WO-2005035500-A2 THERAPEUTIC AGENTS USEFUL FOR TREATING PAIN EURO-CELTIQUE S.A. (LU) 2005-04-21 WO disclosed
EP-1519751-A2 COMPOSITIONS COMPRISING PANTHETINE FOR THE TREATMENT OF DYSLIPIDEMIA Esperion Therapeutics Inc. (US) 2005-04-06 EP disclosed
WO-2004004774-A2 COMPOSITIONS COMPRISING PANTHETINE FOR THE TREATMENT OF DYSLIPIDEMIA ESPERION THERAPEUTICS, INC. (US) 2004-01-15 WO disclosed
US-6340702-B1 SIALIDASE INHIBITORS; ANTIVIRAL COMPOUNDS SANKYO COMPANY, LIMITED (JP) 2002-01-22 US disclosed
CN-1152908-A Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them BASF AG (DE) 1997-06-25 CN disclosed