SCHEMBL4942268

SCHEMBL4942268

NCC(=O)Nc1ccc(Cl)c(NC2=NC(=O)/C(=C/c3ccc4ncccc4c3)S2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
DYRK3 O43781 3/20 0.42
NPC1 O15118 2/20 0.40
PIK3CD O00329 1/20 0.40
PIM1 P11309 1/20 0.40
CSNK2A2 P19784 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CG P48736 1/20 0.40
CLK1 P49759 1/20 0.40
CLK3 P49761 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
DYRK1A Q13627 1/20 0.40
HASPIN Q8TF76 1/20 0.40
DYRK2 Q92630 1/20 0.40
MYLK2 Q9H1R3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2993651 0.92 TSHR (0.42) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2993647 0.92 TSHR (0.42) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL4946166 0.91 DYRK3 (0.42) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL4947101 0.91 DYRK3 (0.42) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2989471 0.90 DYRK3 (0.47) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2989478 0.90 DYRK3 (0.47) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2993503 0.90 ALDH1A1 (0.40) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2993505 0.90 ALDH1A1 (0.40) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2997009 0.90 DYRK3 (0.41) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10
SCHEMBL2996091 0.90 NOTUM (0.43) ALDH1A1CYP3A4CYP1A2TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885362-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-02-13 EP claimed
WO-2006127458-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-30 WO claimed
EP-1885362-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-02-13 EP disclosed
WO-2006127458-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-30 WO disclosed