SCHEMBL4942826

SCHEMBL4942826

O=C1CC(C(F)(F)F)=CN=C1n1nnc(-c2cc(OCc3ccccc3)c(OCc3ccccc3)c([N+](=O)[O-])c2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.35
ABCB1 P08183 1/20 0.34
PTPN1 P18031 4/20 0.33
PTPN6 P29350 3/20 0.33
PTPN2 P17706 2/20 0.33
GRM5 P41594 2/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
CTSV O60911 2/20 0.31
CTSL P07711 2/20 0.31
CYP19A1 P11511 2/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
PTGES O14684 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3592541 0.80 POLB (0.39) POLBPTPN1PTPN6PTPN2GRM5
SCHEMBL1447746 0.78 PTPN1 (0.37) POLBABCB1PTPN1PTPN6PTPN2
SCHEMBL1447254 0.68 MRGPRX4 (0.44) CYP19A1CYP11B1CYP11B2
SCHEMBL1447240 0.66 POLB (0.46) POLBNPC1MAPTRAB9A
SCHEMBL27717189 0.65 MAPT (0.48) PTPN1PTPN6PTPN2NPC1MAPT
SCHEMBL1447215 0.65 POLB (0.43) POLBNPC1MAPTRAB9A
SCHEMBL1447293 0.65 POLB (0.49) POLBNPC1MAPTRAB9AHTR1A
SCHEMBL4948554 0.64 EIF4E (0.38) POLBABCB1NPC1MAPTRAB9A
SCHEMBL3581595 0.64 POLB (0.47) POLBNPC1MAPTRAB9A
SCHEMBL8077523 0.63 CYP19A1 (0.55) POLBMAPTCTSVCTSLCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed