SCHEMBL4948554

SCHEMBL4948554

O=C1CC=NC(C(F)(F)F)=C1c1nc(-c2cc(OCc3ccccc3)c(OCc3ccccc3)c([N+](=O)[O-])c2)cs1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 10/20 0.38
PIN1 Q13526 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
MAPT P10636 2/20 0.33
ABCB1 P08183 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PTGER1 P34995 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
RECQL P46063 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3590056 0.80 EIF4E (0.44) EIF4ECYP19A1CYP11B1CYP11B2
SCHEMBL1446807 0.78 EIF4E (0.42) EIF4ECYP19A1CYP11B1CYP11B2
SCHEMBL4947748 0.74 PTGES (0.38) PIN1CYP19A1MAPTABCB1KDM4E
SCHEMBL4948714 0.70 MAPT (0.37) MAPTABCB1LMNASMN1; SMN2POLB
SCHEMBL28776335 0.69 EIF4E (0.46) EIF4ECYP19A1CYP11B1CYP11B2MAPT
SCHEMBL4942728 0.67 SMN1; SMN2 (0.37) CYP19A1MAPTABCB1KDM4ESMN1; SMN2
SCHEMBL21199376 0.66 KDM4E (0.49) CYP19A1MAPTKDM4ENPC1LMNA
SCHEMBL3581708 0.65 TUBB4A (0.41) PIN1CYP19A1CYP11B1CYP11B2NPC1
SCHEMBL3581595 0.64 POLB (0.47) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL4942826 0.64 POLB (0.35) CYP19A1CYP11B1CYP11B2MAPTABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed