SCHEMBL4943902

SCHEMBL4943902

COc1cc(C(=O)C2=C(C(F)(F)F)N=CCC2=O)ccc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 1/20 0.51
SLC22A8 Q8TCC7 1/20 0.51
MEN1 O00255 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
HTT P42858 1/20 0.44
CXCL12 P48061 1/20 0.40
HSD17B2 P37059 1/20 0.40
CYP1A2 P05177 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
BLM P54132 1/20 0.39
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
APP P05067 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7367773 0.71 SLC22A6 (0.73) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL15814046 0.71 SLC22A6 (1.00) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL28911163 0.67 SLC22A6 (0.77) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL7365546 0.67 SLC22A6 (0.60) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL7369813 0.67 SLC22A6 (0.89) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL7374991 0.66 SLC22A6 (0.80) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL3586390 0.66 SLC22A6 (0.55) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL28149671 0.66 SLC22A6 (0.86) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL30355063 0.66 SLC22A6 (0.86) SLC22A6SLC22A8MEN1RAB9AKMT2A
SCHEMBL3853620 0.65 MEN1 (0.72) SLC22A6SLC22A8MEN1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed