SCHEMBL4943941

SCHEMBL4943941

CNS(=O)(=O)N(C)c1c2c(c(O)c3ncccc13)C(=O)N(Cc1ccc(F)cc1)C2.CNS(=O)(=O)N(C)c1c2c(c(O[Si](C(C)C)(C(C)C)C(C)C)c3ncccc13)C(=O)N(Cc1ccc(F)cc1)C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
LMNA P02545 1/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTGER4 P35408 9/20 0.32
CNR2 P34972 3/20 0.32
COMT P21964 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CACNA2D1 P54289 1/20 0.31
CNR1 P21554 1/20 0.31
IDH1 O75874 1/20 0.31
TBXA2R P21731 1/20 0.31
PTGFR P43088 1/20 0.31
PTGER3 P43115 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5647884 0.96 CACNA2D1 (0.33) KDM4EPTGER4CACNA2D1IDH1TBXA2R
SCHEMBL4750609 0.91 KDM4E (0.38) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL4653390 0.88 PTGER4 (0.32) KDM4EPTGER4L3MBTL1CACNA2D1IDH1
SCHEMBL4691035 0.84 KDM4E (0.38) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL12378080 0.83 KDM4E (0.37) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL29390607 0.83 KDM4E (0.39) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL4652222 0.83 KDM4E (0.39) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL4693753 0.82 KDM4E (0.39) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL4694673 0.82 KDM4E (0.39) KDM4ELMNAHSP90AA1MAPTHTT
SCHEMBL12378084 0.82 KDM4E (0.38) KDM4ELMNAHSP90AA1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888581-A2 HIV-INTEGRASE INHIBITOR COMPOUNDS GILEAD SCIENCES, INC. (US) 2008-02-20 EP disclosed
WO-2006125048-A2 HIV-INTEGRASE INHIBITOR COMPOUNDS GILEAD SCIENCES, INC. (US) 2006-11-23 WO disclosed