SCHEMBL4944904

SCHEMBL4944904

CCCS(=O)(=O)c1cc(Cl)cc2c(Nc3cncc(Cl)c3)c(C(N)=O)cnc12

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 7/20 0.43
PDE4B Q07343 12/20 0.42
TP53 P04637 1/20 0.40
PDE4A P27815 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4947745 0.93 CSF1R (0.45) CSF1RPDE4BTP53PDE4APDE4C
SCHEMBL2478118 0.86 PDE4B (0.45) CSF1RPDE4B
SCHEMBL4950086 0.86 PDE4B (0.42) CSF1RPDE4BTP53PDE4APDE4C
SCHEMBL4951706 0.85 CSF1R (0.45) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL2477404 0.85 PDE4B (0.51) CSF1RPDE4BTP53
SCHEMBL4947634 0.85 CSF1R (0.45) CSF1RPDE4BPDE4APDE4CPDE4D
SCHEMBL5588644 0.82 PDE4B (0.46) CSF1RPDE4BTP53
SCHEMBL1276075 0.81 PDE4B (0.41) CSF1RPDE4B
SCHEMBL1275855 0.81 PDE4B (0.47) CSF1RPDE4B
SCHEMBL2509132 0.80 PDE4B (0.53) CSF1RPDE4BTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed