SCHEMBL4946444

SCHEMBL4946444

Cn1cc(C(=O)Nc2cc(Cl)ccc2Cl)c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.58
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
RAB9A P51151 2/20 0.53
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
NR4A2 P43354 1/20 0.50
ALDH1A1 P00352 3/20 0.49
MITF O75030 1/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
NPC1 O15118 1/20 0.48
POLB P06746 1/20 0.47
HTT P42858 2/20 0.46
HPGD P15428 2/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.46
GSK3B P49841 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91608 0.84 MAOB (0.54) MAOBKMT2AMEN1RAB9AHDAC1
SCHEMBL5684527 0.83 MAOB (0.53) MAOBKMT2AMEN1RAB9ANR4A2
SCHEMBL92369 0.82 RAB9A (0.64) MAOBKMT2AMEN1RAB9AHDAC1
SCHEMBL91603 0.81 MAOB (0.51) MAOBKMT2AMEN1RAB9ANR4A2
SCHEMBL4811502 0.81 MAOB (0.84) MAOBKMT2AMEN1RAB9ANR4A2
SCHEMBL28749578 0.80 MAOB (0.50) MAOBKMT2AMEN1RAB9ANR4A2
SCHEMBL71040 0.79 ITGB1 (0.57) MAOBKMT2AHDAC1HDAC6NR4A2
SCHEMBL27596557 0.79 ITGB1 (0.52) MAOBKMT2AMEN1RAB9AHDAC1
SCHEMBL12861707 0.78 MAOB (0.48) MAOBKMT2AMEN1HDAC1HDAC6
SCHEMBL12861701 0.78 HDAC1 (0.48) MAOBKMT2AHDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed
EP-1961750-A1 VLA-4 INHIBITORY DRUG Daiichi Sankyo Company, Limited (JP) 2008-08-27 EP disclosed