SCHEMBL4947754

SCHEMBL4947754

CC(C)C[C@H](N)C(=O)Nc1ccc(Cl)c(NC2=NC(=O)/C(=C/c3ccc4ncccc4c3)S2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CIT O14578 6/20 0.41
DYRK3 O43781 2/20 0.39
ALDH1A1 P00352 1/20 0.38
AAK1 Q2M2I8 7/20 0.38
CISD1 Q9NZ45 1/20 0.37
PIK3CD O00329 1/20 0.37
PIM1 P11309 1/20 0.37
CSNK2A2 P19784 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CG P48736 1/20 0.37
CLK1 P49759 1/20 0.37
CLK3 P49761 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
DYRK1A Q13627 1/20 0.37
HASPIN Q8TF76 1/20 0.37
DYRK2 Q92630 1/20 0.37
MYLK2 Q9H1R3 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
STK17A Q9UEE5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4944544 0.92 DYRK3 (0.41) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2996481 0.90 DYRK3 (0.42) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2996479 0.90 DYRK3 (0.42) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2999961 0.89 CDK1 (0.44) CITDYRK3ALDH1A1CISD1PIK3CD
SCHEMBL2999956 0.89 CDK1 (0.44) CITDYRK3ALDH1A1CISD1PIK3CD
SCHEMBL2993505 0.88 ALDH1A1 (0.40) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2993503 0.88 ALDH1A1 (0.40) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2997008 0.88 DYRK3 (0.41) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2997009 0.88 DYRK3 (0.41) DYRK3ALDH1A1CISD1PIK3CDPIM1
SCHEMBL2993877 0.86 NPC1 (0.41) DYRK3CISD1PIK3CDPIM1CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885362-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-02-13 EP claimed
WO-2006127458-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-30 WO claimed