SCHEMBL4947801

SCHEMBL4947801

N=CCN1CCC(c2cc(C(N)=O)on2)CC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCD O00767 3/20 0.41
DRD2 P14416 3/20 0.39
DRD4 P21917 3/20 0.39
DRD3 P35462 3/20 0.39
CCR5 P51681 1/20 0.36
SMYD3 Q9H7B4 2/20 0.36
PSMB8 P28062 1/20 0.35
PSMB9 P28065 1/20 0.35
PSMB5 P28074 1/20 0.35
PDE2A O00408 1/20 0.32
ACHE P22303 1/20 0.31
SCD5 Q86SK9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3989771 0.83 SCD (0.44) SCDDRD2DRD4DRD3CCR5
SCHEMBL4149188 0.79 SCD (0.44) SCDDRD2DRD4DRD3SMYD3
SCHEMBL3990440 0.79 SCD (0.50) SCDDRD2DRD4DRD3SMYD3
SCHEMBL3984724 0.79 DRD2 (0.51) SCDDRD2DRD4DRD3ACHE
SCHEMBL3989997 0.77 SCD (0.48) SCDDRD2DRD4DRD3SMYD3
SCHEMBL21317604 0.75 PSMB8 (0.50) SCDSMYD3PSMB8PSMB9PSMB5
SCHEMBL30489440 0.75 PSMB8 (0.50) SCDSMYD3PSMB8PSMB9PSMB5
SCHEMBL3983823 0.75 SCD (0.55) SCDACHESCD5
SCHEMBL3981678 0.73 HRH4 (0.41) SCDSMYD3PSMB8PSMB9PSMB5
SCHEMBL4949165 0.68 SMN1; SMN2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893572-A2 FACTOR XA INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-03-05 EP claimed
WO-2006002099-A2 FACTOR XA INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-01-05 WO claimed
EP-1893572-A2 FACTOR XA INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-03-05 EP disclosed
WO-2006002099-A2 FACTOR XA INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-01-05 WO disclosed