SCHEMBL4948258

SCHEMBL4948258

N#Cc1cnc2sc(/C=C/C(=O)O)cc2c1Cl

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 18/20 0.43
PRKCD Q05655 17/20 0.43
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
LYN P07948 1/20 0.41
HCK P08631 1/20 0.41
SRC P12931 1/20 0.41
PRKCH P24723 1/20 0.41
PRKCE Q02156 1/20 0.41
SLC22A12 Q96S37 1/20 0.35
PLAU P00749 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4948267 1.00 PRKCQ (0.43) PRKCQPRKCDLCKFYNLYN
SCHEMBL4948103 0.81 CYP2A6 (0.36) PRKCQPRKCDLCKFYNLYN
SCHEMBL4909510 0.80 RAB9A (0.34) PRKCQPRKCDSRCSLC22A12PLAU
SCHEMBL4904376 0.80 RAB9A (0.34) PRKCQPRKCDSRCSLC22A12PLAU
SCHEMBL4947800 0.79 SLC22A12 (0.40) SLC22A12
SCHEMBL4947940 0.73 CSNK1A1 (0.36) PRKCQPRKCDLYN
SCHEMBL4950643 0.72 PRKCQ (0.79) PRKCQPRKCDLCKFYNLYN
SCHEMBL4950656 0.72 PRKCQ (0.79) PRKCQPRKCDLCKFYNLYN
SCHEMBL3993667 0.71 CSNK1A1 (0.34) PRKCQPRKCDLYNSRC
SCHEMBL3996010 0.71 CYP2A6 (0.35) PRKCQPRKCDLYNSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937690-A1 THIENO[2,3-B]PYRIDINE-5-CARBONITRILES AS PROTEIN KINASE INHIBITORS Wyeth a Corporation of the State of Delaware (US) 2008-07-02 EP disclosed
US-20070082880-A1 Thieno [2,3-B] pyridine-5-carbonitriles as protein kinase inhibitors WYETH 2007-04-12 US disclosed
WO-2007038519-A1 THIENO[2,3-B]PYRIDINE-5-CARBONITRILES AS PROTEIN KINASE INHIBITORS WYETH (US) 2007-04-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070082880-A1 Thieno [2,3-B] pyridine-5-carbonitriles as protein kinase inhibitors MAP4K2, CNKSR1, MAP3K1 PRKCQ 286/4885PRKCD 356/4885LCK 107/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.