SCHEMBL4948407

SCHEMBL4948407

Cc1c(Cl)c(C)[n+]([O-])c(Br)c1/C=C(/C#N)c1cc(O)c(O)c([N+](=O)[O-])c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 6/20 0.46
FTO Q9C0B1 7/20 0.45
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
RECQL P46063 1/20 0.40
KMT2A Q03164 1/20 0.40
TTR P02766 2/20 0.38
ABCC3 O15438 1/20 0.37
ABCC4 O15439 1/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
NR3C1 P04150 1/20 0.37
PGR P06401 1/20 0.37
HTR1A P08908 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
RARB P10826 1/20 0.37
SLC6A2 P23975 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4948470 0.91 FTO (0.45) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL4943899 0.83 FTO (0.47) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL1447179 0.81 FTO (0.53) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL1447177 0.81 FTO (0.53) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL4946977 0.79 FTO (0.47) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL1446997 0.77 TTR (0.53) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL4946946 0.77 FTO (0.47) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL1447039 0.75 FTO (0.43) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL1446733 0.74 FTO (0.54) COMTFTOMEN1ALDH1A1MAPT
SCHEMBL1446730 0.74 FTO (0.54) COMTFTOMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed