Propyne

Propyne

SCHEMBL4948649

C#CC.Cc1onc(-c2ccccc2)c1C(=O)c1c[nH]c(C(=O)O)c1

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
GAA P10253 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 4/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 1/20 0.46
POLB P06746 2/20 0.45
TSHR P16473 2/20 0.45
MAPK1 P28482 2/20 0.45
ALOX15 P16050 1/20 0.45
ALOX12 P18054 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3977220 0.94 HTT (0.65) HTTSMN1; SMN2GAAKMT2AMEN1
Propyne SCHEMBL4947242 0.86 SMN1; SMN2 (0.48) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL27715447 0.85 HTT (0.56) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL3975278 0.85 HTT (0.55) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL4948655 0.84 HTT (0.58) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL3980271 0.84 HTT (0.70) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL3978785 0.84 SMN1; SMN2 (0.54) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL3973666 0.84 HTT (0.54) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL3976793 0.84 HTT (0.54) HTTSMN1; SMN2GAAKMT2AMEN1
SCHEMBL3975091 0.83 HTT (0.54) HTTSMN1; SMN2GAAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931661-B1 ISOXAZOLO DERIVATIVES AS GABA A ALPHA5 INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-11-19 EP disclosed