SCHEMBL4948655

SCHEMBL4948655

C#CCOC(=O)c1cc(C(=O)c2c(-c3ccccc3)noc2C)c[nH]1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
POLB P06746 1/20 0.51
ALOX15 P16050 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
LMNA P02545 3/20 0.48
ALDH1A1 P00352 2/20 0.48
NPC1 O15118 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
GAA P10253 1/20 0.46
ATM Q13315 1/20 0.45
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4947254 0.88 HTT (0.45) HTTSMN1; SMN2POLBALOX15TSHR
SCHEMBL3982594 0.85 SMN1; SMN2 (0.63) HTTSMN1; SMN2POLBALOX15TSHR
Propyne SCHEMBL4948649 0.84 HTT (0.60) HTTSMN1; SMN2POLBALOX15TSHR
SCHEMBL3980271 0.84 HTT (0.70) HTTSMN1; SMN2POLBTSHRLMNA
SCHEMBL14546677 0.83 HTT (0.61) HTTSMN1; SMN2POLBALOX15TSHR
SCHEMBL3977220 0.83 HTT (0.65) HTTSMN1; SMN2POLBALOX15TSHR
SCHEMBL3981169 0.82 HTT (0.56) HTTSMN1; SMN2POLBALOX15TSHR
SCHEMBL3980161 0.78 HTT (0.60) HTTSMN1; SMN2POLBALOX15TSHR
SCHEMBL3977188 0.78 SMN1; SMN2 (0.55) HTTSMN1; SMN2POLBTSHRLMNA
SCHEMBL3983004 0.78 HTT (0.65) HTTSMN1; SMN2POLBALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931661-B1 ISOXAZOLO DERIVATIVES AS GABA A ALPHA5 INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-11-19 EP disclosed