SCHEMBL4949963

SCHEMBL4949963

CC(C)(C)S(=O)(=O)c1cccc2c(Nc3cncc(Cl)c3)c(C(N)=O)cnc12

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 15/20 0.48
CSF1R P07333 3/20 0.46
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4951706 0.88 CSF1R (0.45) PDE4BCSF1R
SCHEMBL4950378 0.86 PDE4B (0.42) PDE4BCSF1R
SCHEMBL2480619 0.83 PDE4B (0.46) PDE4BCSF1R
SCHEMBL2478780 0.82 PDE4B (0.52) PDE4BCSF1R
SCHEMBL4951341 0.81 PDE4B (0.66) PDE4BMAPT
SCHEMBL2481344 0.81 PDE4B (0.63) PDE4BCSF1R
SCHEMBL4948633 0.80 PDE4B (0.67) PDE4BCSF1RMAPT
SCHEMBL4949957 0.80 PDE4B (0.43) PDE4BCSF1R
SCHEMBL4949242 0.78 PDE4B (0.48) PDE4BCSF1R
SCHEMBL4947745 0.78 CSF1R (0.45) PDE4BCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed