SCHEMBL4948633

SCHEMBL4948633

CS(=O)(=O)c1cccc2c(Nc3cccc(Cl)c3)c(C(N)=O)cnc12

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 14/20 0.67
CSF1R P07333 2/20 0.58
MAPT P10636 1/20 0.52
LRRK2 Q5S007 1/20 0.48
EGFR P00533 1/20 0.47
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4951411 0.88 CSF1R (0.58) PDE4BCSF1RLRRK2
SCHEMBL4948607 0.86 PDE4B (0.68) PDE4B
SCHEMBL4952296 0.85 PDE4B (0.72) PDE4BCSF1RLRRK2
SCHEMBL4948799 0.83 PDE4B (0.56) PDE4BCSF1RLRRK2
SCHEMBL4948831 0.83 PDE4B (0.56) PDE4BCSF1RLRRK2
SCHEMBL4950158 0.82 PDE4B (0.73) PDE4BCSF1REGFR
SCHEMBL1275575 0.80 PDE4B (1.00) PDE4BCSF1R
SCHEMBL4949963 0.80 PDE4B (0.48) PDE4BCSF1RMAPT
SCHEMBL4952544 0.80 PDE4B (0.70) PDE4BCSF1RLRRK2
SCHEMBL4949063 0.77 CSF1R (0.56) PDE4BCSF1RLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed