SCHEMBL4950798

SCHEMBL4950798

COc1ccc2c(c1)OC1(C=C2c2ccccc2)CCN(CC(=O)O)CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 11/20 0.47
KCNH2 Q12809 9/20 0.47
OPRK1 P41145 2/20 0.42
S1PR5 Q9H228 4/20 0.42
S1PR1 P21453 2/20 0.42
GPR55 Q9Y2T6 4/20 0.41
CNR2 P34972 3/20 0.41
S1PR3 Q99500 2/20 0.40
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7175052 0.99 OPRD1 (0.47) OPRD1KCNH2OPRK1S1PR5S1PR1
SCHEMBL4281185 0.90 OPRD1 (0.46) OPRD1KCNH2OPRK1GPR55CNR2
Hydrochloric Acid SCHEMBL4276817 0.88 OPRD1 (0.61) OPRD1KCNH2OPRK1CYP2D6
Hydrochloric Acid SCHEMBL4269370 0.87 OPRD1 (0.49) OPRD1KCNH2OPRK1CYP2D6
Hydrochloric Acid SCHEMBL4284815 0.85 OPRD1 (0.47) OPRD1KCNH2OPRK1CYP2D6
SCHEMBL4273935 0.84 OPRD1 (0.54) OPRD1KCNH2OPRK1CNR2CYP2D6
Hydrochloric Acid SCHEMBL4276512 0.84 OPRD1 (0.46) OPRD1KCNH2OPRK1S1PR5S1PR1
Hydrochloric Acid SCHEMBL4284761 0.83 OPRD1 (0.46) OPRD1KCNH2OPRK1CYP2D6
Hydrochloric Acid SCHEMBL4270071 0.81 OPRD1 (0.55) OPRD1KCNH2OPRK1CYP2D6
Hydrochloric Acid SCHEMBL4272464 0.80 OPRD1 (0.52) OPRD1KCNH2OPRK1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1232160-B1 SPIRO(2H-1-BENZOPYRAN-2,4'-PIPERIDINE)DERIVATES AS GLYCINE TRANSPORT INHIBITORS ORGANON NV (NL) 2008-06-18 EP disclosed