SCHEMBL4951273

SCHEMBL4951273

N#C/C(=C/c1cc(C(F)(F)F)c[n+]([O-])c1)c1cc(O)c(O)c([N+](=O)[O-])c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 5/20 0.50
TTR P02766 3/20 0.47
COMT P21964 2/20 0.45
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
RECQL P46063 2/20 0.45
KMT2A Q03164 2/20 0.45
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
KDM4E B2RXH2 1/20 0.38
GMNN O75496 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
THRB P10828 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1447201 0.88 FTO (0.58) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL1447198 0.88 FTO (0.58) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL4954976 0.81 FTO (0.52) FTOTTRCOMTMEN1ALDH1A1
SCHEMBL3590974 0.76 FTO (0.71) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL3590969 0.76 FTO (0.71) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL1447200 0.76 TTR (0.67) TTRCOMTMEN1ALDH1A1MAPT
SCHEMBL4944869 0.75 FTO (0.43) FTOTTRCOMTMEN1ALDH1A1
SCHEMBL1447039 0.75 FTO (0.43) FTOTTRCOMTMEN1ALDH1A1
SCHEMBL1446766 0.75 FTO (0.60) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL1446769 0.75 FTO (0.60) FTOCOMTMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed