SCHEMBL4959417

SCHEMBL4959417

NC(=O)OC(COc1ccc(Cl)cc1)Cn1nnc(I)n1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
LTA4H P09960 7/20 0.43
SLC6A3 Q01959 2/20 0.41
CYP19A1 P11511 1/20 0.40
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4310465 0.81 CYP1A2 (0.49) CYP1A2CYP19A1ALDH1A1KMT2APPARG
SCHEMBL4304641 0.80 CYP1A2 (0.45) CYP1A2LTA4HCYP19A1POLBPPARG
SCHEMBL4311966 0.76 CYP1A2 (0.46) CYP1A2CYP19A1POLBMAPTKMT2A
SCHEMBL4315990 0.75 CYP1A2 (0.45) CYP1A2CYP19A1PPARGPPARA
SCHEMBL4309877 0.69 ALDH1A1 (0.36) CYP1A2CYP19A1ALDH1A1POLBKMT2A
SCHEMBL4314433 0.68 POLB (0.35) CYP1A2ALDH1A1POLBKMT2A
SCHEMBL4309847 0.66 CYP1A2 (0.44) CYP1A2MAPT
SCHEMBL4304481 0.65 POLB (0.35) ALDH1A1POLBKMT2A
SCHEMBL4312614 0.63 KMT2A (0.43) CYP1A2ALDH1A1POLBMAPTKMT2A
SCHEMBL4311700 0.62 POLB (0.43) CYP1A2ALDH1A1POLBMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879873-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK Holdings Co., Ltd. (KR) 2008-01-23 EP disclosed
WO-2006112685-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK HOLDINGS CO., LTD. (KR) 2006-10-26 WO disclosed