SCHEMBL4960028

SCHEMBL4960028

CS(=O)(=O)c1ccc(-c2[nH]nc(CCCO)c2CC2CCCCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.42
PTGS1 P23219 4/20 0.42
GHSR Q92847 1/20 0.35
CCNB2 O95067 2/20 0.34
CDK1 P06493 2/20 0.34
CCNB1 P14635 2/20 0.34
GSK3A P49840 2/20 0.34
GSK3B P49841 2/20 0.34
CCNB3 Q8WWL7 2/20 0.34
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958133 0.89 PTGS2 (0.44) PTGS2PTGS1GHSRCCNB2CDK1
SCHEMBL4957399 0.85 PTGS2 (0.43) PTGS2PTGS1CCNB2CDK1CCNB1
SCHEMBL4959251 0.85 PTGS2 (0.40) PTGS2PTGS1GHSRCCNB2CDK1
SCHEMBL4958756 0.85 PTGS2 (0.44) PTGS2PTGS1GHSRCCNB2CDK1
SCHEMBL4958956 0.83 CCNB2 (0.35) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL6439748 0.83 PTGS2 (0.44) PTGS2PTGS1GHSRKMT2A
SCHEMBL4957579 0.80 PTGS2 (0.48) PTGS2PTGS1GHSRCCNB2CDK1
SCHEMBL6439645 0.79 PTGS2 (0.42) PTGS2PTGS1GHSR
SCHEMBL4957792 0.79 CCNB2 (0.41) PTGS2PTGS1GHSRCCNB2CDK1
SCHEMBL4957380 0.78 PTGS2 (0.41) PTGS2PTGS1CCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP claimed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP claimed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO claimed
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP disclosed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP disclosed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO disclosed