SCHEMBL4963344

SCHEMBL4963344

CCC1(CC)C(=O)N(C(C)C)c2cc3nc(-c4[c]cn(C(N)=O)n4)[nH]c3cc21

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4891843 0.88 AURKA (0.39) AURKAAURKB
SCHEMBL4966344 0.88 AURKA (0.44) AURKAAURKB
SCHEMBL4888268 0.79 AURKA (0.56) AURKAAURKB
SCHEMBL4891866 0.74 PDE4A (0.52) AURKAAURKB
SCHEMBL4822495 0.73 AURKA (0.38) AURKAAURKB
SCHEMBL5952304 0.73 CHEK2 (0.36)
SCHEMBL3578314 0.71 AMY1A (0.42)
SCHEMBL4829089 0.69 SYK (0.39) AURKAAURKB
SCHEMBL5953327 0.69 SYK (0.43)
SCHEMBL4822663 0.69 PDPK1 (0.35) AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879894-A1 AMINOPYRAZOLE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2008-01-23 EP disclosed
WO-2006108489-A1 AMINOPYRAZOLE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2006-10-19 WO disclosed