SCHEMBL4963422

SCHEMBL4963422

Nc1nc2nc[nH]c2c(=O)n1Cc1ccc(Br)s1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.40
PDE4A P27815 3/20 0.37
PDE4B Q07343 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
PDPK1 O15530 1/20 0.36
GDA Q9Y2T3 1/20 0.36
MGMT P16455 2/20 0.35
ALDH1A1 P00352 2/20 0.35
DPP4 P27487 1/20 0.35
ADORA2B P29275 3/20 0.35
ADORA2A P29274 2/20 0.35
KDM4E B2RXH2 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PIN1 Q13526 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3300188 0.85 PNP (0.40) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL9434524 0.85 PNP (0.40) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL5084763 0.82 MGMT (0.52) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL8208746 0.81 PNP (0.45) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL4962859 0.81 PDE4A (0.53) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL4963405 0.81 MGMT (0.35) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL3310277 0.80 PNP (0.50) PNPPDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL18605981 0.80 PDE4A (0.53) PNPPDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL17186468 0.79 PNP (0.49) PNPPDE4APDE4BPDE4CPDE4D
SCHEMBL4967495 0.78 PNP (0.38) PNPPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4054057-B2 2008-02-27 JP claimed
EP-0702683-B1 06-SUBSTITUTED GUANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN TREATING TUMOUR CELLS CANCER REC TECH LTD (GB) 2003-09-17 EP claimed
WO-1994029312-A1 O6-SUBSTITUTED GUANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN TREATING TUMOUR CELLS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1994-12-22 WO claimed
EP-0702683-B1 06-SUBSTITUTED GUANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN TREATING TUMOUR CELLS CANCER REC TECH LTD (GB) 2003-09-17 EP disclosed
WO-1994029312-A1 O6-SUBSTITUTED GUANINE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN TREATING TUMOUR CELLS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1994-12-22 WO disclosed